WebAug 7, 2024 · The carboxylation of sp3-hybridized C–H bonds with CO2 is a challenging transformation. Herein, we report a visible-light-mediated carboxylation of benzylic C–H bonds with CO2 into 2-arylpropionic acids under metal-free conditions. Photo-oxidized triisopropylsilanethiol was used as the hydrogen atom transfer catalyst to afford a … WebJul 11, 2024 · The carboxylation of sp 3-hybridized C–H bonds with CO 2 is a challenging transformation. Herein, we report a visible-light-mediated carboxylation of benzylic C–H …
Burkhard KÖNIG Professor (Full) Universität Regensburg, …
WebDec 18, 2024 · A photoinduced carboxylation reaction of benzylic and aliphatic C-H bonds with CO 2 is developed. Toluene derivatives capture gaseous CO 2 at the benzylic position … WebAug 1, 2024 · (Hetero)benzylic C–H bonds are prevalent in medicinal and bioactive molecules, and these positions are prone to oxidation catalyzed by enzymes during metabolization. 68 Selective functionalization of those C–H bonds could potentially tune the metabolic stability of drugs and regulate the bioactivity of lead compounds or drug … e650i-a2 wireless speakers for outdoor
Mechanistic study on the photo carboxylation of benzylic C-H bonds …
WebThe C−H substrate is used as limiting reagent with only a small excess of the unactivated amide or carbamate nucleophile. The enantioselective intermolecular dehydrogenative C−N bond formation is enabled by a combination of a chiral copper catalyst, a photocatalyst, and an oxidant, and it takes place under mild conditions, which allow for a ... WebWith a deep understanding of photo-introduced HAT, it was established that the bond dissociation energy (BDE) of the benzylic C–H bond is around 84–90 kcal/mol (for example, BDE in a benzylic C–H bond of toluene is 88 kcal/mol), which is not easy to abstract by the formed bromide radical (87 kcal/mol). WebNov 25, 2024 · A highly efficient carboxylation of benzyl alcohol derivatives with CO2using a palladium/iridium dual catalyst under visible-light irradiation was developed. A wide range of benzyl alcohol derivatives could be employed to provide benzylic carboxylic acids in moderate to high yields. cs go download for windows 10 free edition